Brief Information of the Compound and Protein
Compound Name
US8835444, 3.6
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PubChem ID
SID: 125259376
Canonical SMILES
Cc1cc(nn1C[C@H]1CC[C@@H](CC1)NC(=O)c1cc(Cl)cnc1C)-c1cccnc1
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Compound Formula C23H26ClN5O
Compound Structure
Protein Name
Corticotropin-releasing factor receptor 2
Protein Classification
Membrane receptor
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Family B G protein-coupled receptor
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Peptide receptor (family B GPCR)
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Corticotropin releasing factor receptor
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Corticotropin releasing factor receptor
Uniprot ID
Q13324
Gene Name
CRHR2
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
IC50 = 3737 nM
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