Brief Information of the Compound and Protein
Compound Name
US8722896, N-[(+/-)-2-Methyl-3-(indol- 4ylmethyl)aminopropanoyl]- (+/-)-valyl-(3,4-dihydro-2H-1,5- benzodioxepin-7- ylmethyl)amide
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PubChem ID
CID: 58080642
Canonical SMILES
CC(C)C(NC(=O)C(C)CNCc1cccc2[nH]ccc12)C(=O)NCc1ccc2OCCCOc2c1
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Compound Formula C28H36N4O4
Compound Structure
Protein Name
Prokineticin receptor 2
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Peptide growth factor receptor (family A GPCR)
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Prokineticin receptor
Uniprot ID
G3H407
Gene Name
PROKR2
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 248 nM
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