Brief Information of the Compound and Protein
Compound Name
US8722896, (-)-(3R)-1-(Indol-7-ylmethyl)-N- (6-chloro-2,3,4,5-tetrahydro-1- benzoxepin-8-ylmethyl)-N- isobutylpyrrolidine-3- carboxamide
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PubChem ID
CID: 58080429
Canonical SMILES
CC(C)CN(Cc1cc(Cl)c2CCCCOc2c1)C(=O)C1CCN(Cc2cccc3cc[nH]c23)C1
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Compound Formula C29H36ClN3O2
Compound Structure
Protein Name
Prokineticin receptor 2
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Peptide growth factor receptor (family A GPCR)
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Prokineticin receptor
Uniprot ID
G3H407
Gene Name
PROKR2
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 82 nM
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