Brief Information of the Compound and Protein
Compound Name
US8722896, (+/-)-2-Methyl-3-(indol-4- ylmethylamino)-N-(9-chloro- 3,4-dihydro-2H-1,5- benzodioxepin-7-ylmethyl)-N- propylpanamide
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PubChem ID
CID: 58080639
Canonical SMILES
CCCN(Cc1cc(Cl)c2OCCCOc2c1)C(=O)C(C)CNCc1cccc2[nH]ccc12
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Compound Formula C26H32ClN3O3
Compound Structure
Protein Name
Prokineticin receptor 2
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Peptide growth factor receptor (family A GPCR)
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Prokineticin receptor
Uniprot ID
G3H407
Gene Name
PROKR2
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 15.8 nM
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   LI
   LO
   TS