Brief Information of the Compound and Protein
Compound Name
7-(5-chloro-2,3-dihydroindol-1-yl)-9-methoxy-4-(pyridin-3-ylmethyl)-3,5-dihydro-2H-1,4-benzoxazepine
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PubChem ID
CID: 122180284
Canonical SMILES
COc1cc(cc2CN(Cc3cccnc3)CCOc12)N1CCc2cc(Cl)ccc12
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Compound Formula C24H24ClN3O2
Compound Structure
Protein Name
Prostaglandin E2 receptor EP2 subtype
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Lipid-like ligand receptor (family A GPCR)
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Prostanoid receptor
Uniprot ID
P43116
Gene Name
PTGER2
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000516 ECV-304 Homo sapiens (Human)  2
1
IC50 = 30 nM
   TI
   LI
   LO
   TS
2
IC50 = 60 nM
   TI
   LI
   LO
   TS