Brief Information of the Compound and Protein
Compound Name
(R)-5-((4'-(2-(2-methylpyrrolidin-1-yl)ethyl)biphenyl-4-yl)methyl)-1H-tetrazole
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PubChem ID
CID: 78321037
Canonical SMILES
C[C@@H]1CCCN1CCc1ccc(-c2ccc(Cc3nnn[nH]3)cc2)cc1
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Compound Formula C21H25N5
Compound Structure
Protein Name
Histamine H3 receptor
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Histamine receptor
Uniprot ID
Q9Y5N1
Gene Name
HRH3
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 0.78 nM
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   LI
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