Brief Information of the Compound and Protein
Compound Name
methyl 1-[4-[4-[2-[(2R)-2-methylpyrrolidin-1-yl]ethyl]phenyl]phenyl]cyclopentane-1-carboxylate
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PubChem ID
CID: 78320398
Canonical SMILES
COC(=O)C1(CCCC1)c1ccc(cc1)-c1ccc(CCN2CCC[C@H]2C)cc1
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Compound Formula C26H33NO2
Compound Structure
Protein Name
Histamine H3 receptor
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Histamine receptor
Uniprot ID
Q9Y5N1
Gene Name
HRH3
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 3.3 nM
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