Brief Information of the Compound and Protein
Compound Name
N-methyl-7-(4-methylsulfonylphenyl)-N-(1-propan-2-ylsulfonylpiperidin-4-yl)thieno[3,2-d]pyrimidin-4-amine
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PubChem ID
CID: 118709767
Canonical SMILES
CC(C)S(=O)(=O)N1CCC(CC1)N(C)c1ncnc2c(csc12)-c1ccc(cc1)S(C)(=O)=O
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Compound Formula C22H28N4O4S3
Compound Structure
Protein Name
Glucose-dependent insulinotropic receptor
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Lipid-like ligand receptor (family A GPCR)
Uniprot ID
Q8TDV5
Gene Name
GPR119
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000026 CHO-K1 Cricetulus griseus (Chinese hamster)  1
1
EC50 = 1200 nM
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