Brief Information of the Compound and Protein
Compound Name
4-[[(3S,4R)-4-(4-chlorophenyl)-1-(2,2,2-trifluoroethyl)piperidin-3-yl]methoxy]-2,5-difluoro-N-(1,2,4-thiadiazol-5-yl)benzenesulfonamide
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PubChem ID
CID: 89545670
Canonical SMILES
Fc1cc(c(F)cc1OC[C@@H]1CN(CC(F)(F)F)CC[C@H]1c1ccc(Cl)cc1)S(=O)(=O)Nc1ncns1
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Compound Formula C22H20ClF5N4O3S2
Compound Structure
Protein Name
Sodium channel protein type 5 subunit alpha
Protein Classification
Ion channel
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Voltage-gated ion channel
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Voltage-gated sodium channel
Uniprot ID
Q14524
Gene Name
SCN5A
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 2600 nM
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