Brief Information of the Compound and Protein
Compound Name
2,5-difluoro-4-[[(3R,4R)-3-(4-fluorophenyl)piperidin-4-yl]methoxy]-N-(1,2,4-thiadiazol-5-yl)benzenesulfonamide
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PubChem ID
CID: 89556066
Canonical SMILES
Fc1ccc(cc1)[C@@H]1CNCC[C@H]1COc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1
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Compound Formula C20H19F3N4O3S2
Compound Structure
Protein Name
Sodium channel protein type 5 subunit alpha
Protein Classification
Ion channel
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Voltage-gated ion channel
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Voltage-gated sodium channel
Uniprot ID
Q14524
Gene Name
SCN5A
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 5900 nM
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