Brief Information of the Compound and Protein
Compound Name
methyl (3S)-3-[(3-fluorophenyl)methyl]-10-[4-(trifluoromethyl)phenyl]-1,4,8,12-tetrazatricyclo[7.3.0.02,6]dodeca-2(6),4,7,9,11-pentaene-3-carboxylate
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PubChem ID
CID: 118720421
Canonical SMILES
COC(=O)[C@@]1(Cc2cccc(F)c2)N=Cc2cnc3c(cnn3c12)-c1ccc(cc1)C(F)(F)F
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Compound Formula C24H16F4N4O2
Compound Structure
Protein Name
Glucose-dependent insulinotropic receptor
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Lipid-like ligand receptor (family A GPCR)
Uniprot ID
Q7TQP3
Gene Name
GPR119
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
EC50 = 135 nM
   TI
   LI
   LO
   TS