Brief Information of the Compound and Protein
Compound Name
 Compound Info 
1-[3-[4-(7-hydroxyheptyl)piperidin-1-yl]propyl]-3,4-dihydroquinolin-2-one
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 PubChem ID
CID: 118719927
Canonical SMILES
OCCCCCCCC1CCN(CCCN2C(=O)CCc3ccccc23)CC1
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Compound Formula C24H38N2O2
Compound Structure
Protein Name
 Protein Info 
Muscarinic acetylcholine receptor M4
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Acetylcholine receptor
Uniprot ID
P08173
Gene Name
CHRM4
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  1
1
Ki = 389.05 nM
   TI
   LI
   LO
   TS
CL000025 HEK-293T
 Cell Line Info 
Homo sapiens (Human)  3
1
IC50 = 588.84 nM
   TI
   LI
   LO
   TS
2
IC50 = 794.33 nM
   TI
   LI
   LO
   TS
3
IC50 = 1479.11 nM
   TI
   LI
   LO
   TS