Brief Information of the Compound and Protein
Compound Name
rac-4-(6-((1-Isopropylpiperidin-3-yl)methyl)-7-oxo-5-o-tolyl-6,7-dihydro-2H-pyrazolo[4,3-d]pyrimidin-2-yl)benzonitrile
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PubChem ID
CID: 90665852
Canonical SMILES
Cc1ccccc1-c1nc2cn(-c3ccc(C#N)cc3)nc2c(=O)n1CC1CCCN(C(C)C)C1
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Compound Formula C28H30N6O
Compound Structure
Protein Name
Growth hormone secretagogue receptor type 1
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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GRP-related receptor
Uniprot ID
Q92847
Gene Name
GHSR
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 12 nM
   TI
   LI
   LO
   TS