Brief Information of the Compound and Protein
Compound Name
2-(4-Chlorophenyl)-6-{[(3R)-1-(2-methoxyethyl)piperidin-3-yl]methyl}-5-(2-methylphenyl)[1,3]thiazolo[4,5-d]pyrimidin-7(6H)-one
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PubChem ID
CID: 90665849
Canonical SMILES
COCCN1CCC[C@@H](Cn2c(-c3ccccc3C)nc3nc(-c4ccc(Cl)cc4)sc3c2=O)C1
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Compound Formula C27H29ClN4O2S
Compound Structure
Protein Name
Growth hormone secretagogue receptor type 1
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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GRP-related receptor
Uniprot ID
Q92847
Gene Name
GHSR
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 59 nM
   TI
   LI
   LO
   TS