Brief Information of the Compound and Protein
Compound Name
 Compound Info 
5-cyano-N-[2-(4,4-dimethylcyclohexen-1-yl)-4-[2-(1,1-dioxo-1,4-thiazinan-4-yl)propan-2-yl]phenyl]-1H-imidazole-2-carboxamide
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 PubChem ID
CID: 24874843
SID: 50130110
Canonical SMILES
CC(C)(N1CCS(=O)(=O)CC1)c1ccc(NC(=O)c2ncc([nH]2)C#N)c(c1)C1=CCC(C)(C)CC1
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Compound Formula C26H33N5O3S
Compound Structure
Protein Name
 Protein Info 
Mast/stem cell growth factor receptor Kit
Protein Classification
Enzyme
>
Kinase
>
Protein Kinase
>
TK protein kinase group
>
Tyrosine protein kinase PDGFR family
Uniprot ID
P10721
Gene Name
KIT
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000138 M-07e
 Cell Line Info 
Homo sapiens (Human)  1
1
IC50 = 3300 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 250 nM