Brief Information of the Compound and Protein
Compound Name
 Compound Info 
7-(3,5-dimethyl-1,2-oxazol-4-yl)-8-methoxy-1-[(1R)-1-pyridin-2-ylethyl]-3H-imidazo[4,5-c]quinolin-2-one
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 PubChem ID
CID: 52912189
SID: 123047600
Canonical SMILES
COc1cc2c3n([C@H](C)c4ccccn4)c(=O)[nH]c3cnc2cc1-c1c(C)noc1C
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Compound Formula C23H21N5O3
Compound Structure
Protein Name
 Protein Info 
Bromodomain-containing protein 4
Protein Classification
Epigenetic regulator
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Bromodomain
Uniprot ID
O60885
Gene Name
BRD4
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000174 Raji
 Cell Line Info 
Homo sapiens (Human)  1
1
IC50 = 130 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 18 nM
2 IC50 = 36 nM
3 IC50 = 100 nM
4 IC50 = 107 nM
5 IC50 = 274 nM
6 IC50 = 790 nM
7 IC50 = 794.33 nM
8 Ki = 61 nM
9 Ki = 385 nM