Brief Information of the Compound and Protein
Compound Name
 Compound Info 
3-amino-4,6-dimethyl-N-p-anisyl-thieno[2,3-b]pyridine-2-carboxamide
    Show/Hide
 PubChem ID
CID: 864492
SID: 49691983
Canonical SMILES
COc1ccc(CNC(=O)c2sc3nc(C)cc(C)c3c2N)cc1
    Show/Hide
Compound Formula C18H19N3O2S
Compound Structure
Protein Name
 Protein Info 
Muscarinic acetylcholine receptor M4
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
>
Small molecule receptor (family A GPCR)
>
Monoamine receptor
>
Acetylcholine receptor
Uniprot ID
P08173
Gene Name
CHRM4
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  1
1
EC50 = 495 nM
   TI
   LI
   LO
   TS
CL000026 CHO-K1
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  1
1
EC50 = 620 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 EC50 = 520 nM
2 EC50 = 680 nM