Brief Information of the Compound and Protein
Compound Name
N-[(2R)-3-[4-(4-chloro-2-methylphenoxy)piperidin-1-yl]-2-hydroxypropyl]-5-(trifluoromethyl)-1H-pyrazole-4-carboxamide
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PubChem ID
CID: 59296100
SID: 163526123
Canonical SMILES
Cc1cc(Cl)ccc1OC1CCN(C[C@H](O)CNC(=O)c2cn[nH]c2C(F)(F)F)CC1
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Compound Formula C20H24ClF3N4O3
Compound Structure
Protein Name
Potassium voltage-gated channel subfamily H member 2
Protein Classification
Ion channel
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Voltage-gated ion channel
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Potassium channels
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Voltage-gated potassium channel
Uniprot ID
Q12809
Gene Name
KCNH2
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  2
1
IC50 = 1258.93 nM
   TI
   LI
   LO
   TS
2
IC50 = 3162.28 nM
   TI
   LI
   LO
   TS