Brief Information of the Compound and Protein
Compound Name
 Compound Info 
6-(4-tert-butylphenyl)sulfonyl-7-piperidin-4-yl-2-(trifluoromethyl)-5,11-dihydropyrido[3,2-c][1,5]benzodiazepine
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 PubChem ID
CID: 62707363
SID: 148139024
Canonical SMILES
CC(C)(C)c1ccc(cc1)S(=O)(=O)N1Cc2ccc(nc2Nc2cccc(C3CCNCC3)c12)C(F)(F)F
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Compound Formula C28H31F3N4O2S
Compound Structure
Protein Name
 Protein Info 
Bombesin receptor subtype-3
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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GRP-related receptor
Uniprot ID
P32247
Gene Name
BRS3
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000943 CellSensor NFAT-bla CHO-K1
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  1
1
IC50 = 1.4 nM
   TI
   LI
   LO
   TS
CL000866 HEK293 AequoScreen
 Cell Line Info 
Homo sapiens (Human)  1
1
EC50 = 114 nM
   TI
   LI
   LO
   TS