Brief Information of the Compound and Protein
Compound Name
 Compound Info 
N-(benzylsulfamoyl)-6-[2-(5-bromopyrimidin-2-yl)oxyethoxy]-5-phenylpyrimidin-4-amine
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 PubChem ID
CID: 71455139
SID: 163486220
Canonical SMILES
Brc1cnc(OCCOc2ncnc(NS(=O)(=O)NCc3ccccc3)c2-c2ccccc2)nc1
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Compound Formula C23H21BrN6O4S
Compound Structure
Protein Name
 Protein Info 
Endothelin-1 receptor
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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Endothelin receptor
Uniprot ID
P25101
Gene Name
EDNRA
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  1
1
IC50 = 6.8 nM
   TI
   LI
   LO
   TS