Brief Information of the Compound and Protein
Compound Name
2-[2-(5-fluoropyrimidin-2-yl)ethyl]-N-[[4-fluoro-3-(trifluoromethoxy)phenyl]methyl]-3-oxo-1H-isoindole-1-carboxamide
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PubChem ID
CID: 60201255
SID: 144219081
Canonical SMILES
Fc1cnc(CCN2C(C(=O)NCc3ccc(F)c(OC(F)(F)F)c3)c3ccccc3C2=O)nc1
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Compound Formula C23H17F5N4O3
Compound Structure
Protein Name
Sodium channel protein type 5 subunit alpha
Protein Classification
Ion channel
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Voltage-gated ion channel
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Voltage-gated sodium channel
Uniprot ID
Q14524
Gene Name
SCN5A
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000026 CHO-K1 Cricetulus griseus (Chinese hamster)  1
1
IC50 = 17000 nM
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