Brief Information of the Compound and Protein
Compound Name
4-[[2-[(2R)-4-(5-fluoropyrimidin-2-yl)-2-methylpiperazin-1-yl]pyrimidin-5-yl]oxymethyl]pyridine-3-carbonitrile
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PubChem ID
CID: 51030056
SID: 117690066
Canonical SMILES
C[C@@H]1CN(CCN1c1ncc(OCc2ccncc2C#N)cn1)c1ncc(F)cn1
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Compound Formula C20H19FN8O
Compound Structure
Protein Name
Glucose-dependent insulinotropic receptor
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Lipid-like ligand receptor (family A GPCR)
Uniprot ID
Q8TDV5
Gene Name
GPR119
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000107 HEK293S Homo sapiens (Human)  1
1
EC50 = 63 nM
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   LI
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   TS