Brief Information of the Compound and Protein
Compound Name
N-[3-[1-[3-[1-oxo-4-(2,3,5-trifluorophenyl)phthalazin-2-yl]propyl]piperidin-4-yl]phenyl]acetamide
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PubChem ID
CID: 57397820
SID: 152140722
Canonical SMILES
CC(=O)Nc1cccc(c1)C1CCN(CCCn2nc(-c3cc(F)cc(F)c3F)c3ccccc3c2=O)CC1
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Compound Formula C30H29F3N4O2
Compound Structure
Protein Name
Melanin-concentrating hormone receptor 1
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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MCH receptor
Uniprot ID
Q99705
Gene Name
MCHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
IC50 = 27 nM
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