Brief Information of the Compound and Protein
Compound Name
9-(2-chloro-4-methoxyphenyl)-N-(dicyclopropylmethyl)-2,8-dimethylpurin-6-amine
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PubChem ID
CID: 44545284
SID: 87228152
Canonical SMILES
COc1ccc(c(Cl)c1)-n1c(C)nc2c(NC(C3CC3)C3CC3)nc(C)nc12
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Compound Formula C21H24ClN5O
Compound Structure
Protein Name
Corticotropin-releasing factor receptor 1
Protein Classification
Membrane receptor
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Family B G protein-coupled receptor
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Peptide receptor (family B GPCR)
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Corticotropin releasing factor receptor
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Corticotropin releasing factor receptor
Uniprot ID
P34998
Gene Name
CRHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 12 nM
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