Brief Information of the Compound and Protein
Compound Name
N-[2-[[1-[4-(1H-indol-3-yl)cyclohexyl]azetidin-3-yl]amino]-2-oxoethyl]-3-(trifluoromethyl)benzamide
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PubChem ID
CID: 46946452
SID: 99459352
Canonical SMILES
FC(F)(F)c1cccc(c1)C(=O)NCC(=O)NC1CN(C1)C1CCC(CC1)c1c[nH]c2ccccc12
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Compound Formula C27H29F3N4O2
Compound Structure
Protein Name
Potassium voltage-gated channel subfamily H member 2
Protein Classification
Ion channel
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Voltage-gated ion channel
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Potassium channels
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Voltage-gated potassium channel
Uniprot ID
Q12809
Gene Name
KCNH2
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 2400 nM
   TI
   LI
   LO
   TS