Brief Information of the Compound and Protein
Compound Name
8,12,14-trimethyl-9-(5-methylfuran-2-yl)-17-phenyl-1,8,12,14-tetrazatetracyclo[8.7.0.02,7.011,16]heptadeca-2,4,6,10,16-pentaene-13,15-dione
    Show/Hide
PubChem ID
CID: 53392786
SID: 125321083
Canonical SMILES
CN1C(c2ccc(C)o2)c2n(c(-c3ccccc3)c3c2n(C)c(=O)n(C)c3=O)-c2ccccc12
    Show/Hide
Compound Formula C27H24N4O3
Compound Structure
Protein Name
Cystic fibrosis transmembrane conductance regulator
Protein Classification
Ion channel
>
Other ion channel
>
Chloride channel
>
Cystic fibrosis transmembrane conductance regulator
Uniprot ID
P13569
Gene Name
CFTR
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000259 FRT Rattus norvegicus (Rat)  1
1
IC50 = 1000 nM
   TI
   LI
   LO
   TS