Brief Information of the Compound and Protein
Compound Name
4-bromo-5-((4-(2-methoxyphenyl)piperazin-1-yl)methyl)-1-methyl-2-phenyl-1H-pyrazol-3(2H)-one
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PubChem ID
CID: 54584258
Canonical SMILES
COc1ccccc1N1CCN(Cc2c(Br)c(=O)n(-c3ccccc3)n2C)CC1
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Compound Formula C22H25BrN4O2
Compound Structure
Protein Name
Metabotropic glutamate receptor 2
Protein Classification
Membrane receptor
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Family C G protein-coupled receptor
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Small molecule receptor (family C GPCR)
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Neurotransmitter receptor (family C GPCR)
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Metabotropic glutamate receptor
Uniprot ID
P31421
Gene Name
GRM2
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
EC50 = 891 nM
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