Brief Information of the Compound and Protein
Compound Name
N-[1-[3-(6,7-difluoro-2-oxo-3,4-dihydroquinolin-1-yl)propyl]piperidin-4-yl]-2-(3,4-dimethoxyphenyl)acetamide
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PubChem ID
CID: 44208359
SID: 85208333
Canonical SMILES
COc1ccc(CC(=O)NC2CCN(CCCN3C(=O)CCc4cc(F)c(F)cc34)CC2)cc1OC
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Compound Formula C27H33F2N3O4
Compound Structure
Protein Name
Muscarinic acetylcholine receptor M5
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Acetylcholine receptor
Uniprot ID
P08912
Gene Name
CHRM5
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000051 BHK-21 Mesocricetus auratus (Golden hamster)  1
1
EC50 = 1200 nM
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