Brief Information of the Compound and Protein
Compound Name
(E)-1-[4-(1-azepanylsulfonyl)phenyl]-3-(3,4-dihydroxyphenyl)-2-propen-1-one
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PubChem ID
CID: 5994055
Canonical SMILES
Oc1ccc(\C=C\C(=O)c2ccc(cc2)S(=O)(=O)N2CCCCCC2)cc1O
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Compound Formula C21H23NO5S
Compound Structure
Protein Name
Tyrosine-protein kinase JAK2
Protein Classification
Enzyme
>
Kinase
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Protein Kinase
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TK protein kinase group
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Tyrosine protein kinase JakB family
Uniprot ID
O60674
Gene Name
JAK2
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000077 Ba/F3 Mus musculus (Mouse)  1
1
IC50 = 7505 nM
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