Brief Information of the Compound and Protein
Compound Name
 Compound Info 
(BRL 43694)1-Methyl-1H-indazole-3-carboxylic acid (9-methyl-9-aza-bicyclo[3.3.1]non-3-yl)-amide
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 PubChem ID
CID: 3510
SID: 14874362
Canonical SMILES
CN1C2CCCC1CC(C2)NC(=O)c1nn(C)c2ccccc12
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Compound Formula C18H24N4O
Compound Structure
Protein Name
 Protein Info 
Potassium voltage-gated channel subfamily H member 2
Protein Classification
Ion channel
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Voltage-gated ion channel
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Potassium channels
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Voltage-gated potassium channel
Uniprot ID
Q12809
Gene Name
KCNH2
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293
 Cell Line Info 
Homo sapiens (Human)  1
1
IC50 = 3730 nM
   TI
   LI
   LO
   TS
CL000083 MCF-7
 Cell Line Info 
Homo sapiens (Human)  1
1
IC50 = 3801.89 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 3715.35 nM
2 IC50 = 3801.89 nM