Brief Information of the Compound and Protein
Compound Name
5-[4-[(1,1'-Biphenyl-2-ylcarbonyl)amino]-3-methylbenzoyl]-1-methyl-1,4,5,10-tetrahydropyrazolo[3,4-b][1,5]benzodiazepine
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PubChem ID
CID: 135916059
SID: 92122513
Canonical SMILES
Cc1cc(ccc1NC(=O)c1ccccc1-c1ccccc1)C(=O)N1Cc2cnn(C)c2Nc2ccccc12
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Compound Formula C32H27N5O2
Compound Structure
Protein Name
Vasopressin V2 receptor
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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Vasopressin and oxytocin receptor
Uniprot ID
P30518
Gene Name
AVPR2
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 6.4 nM
   TI
   LI
   LO
   TS