Brief Information of the Compound and Protein
Compound Name
 Compound Info 
4-(2-{3-[(2,2,3,3-tetramethylcyclopropyl)carbonyl]-1H-indol-1-yl}ethyl)morpholine
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 PubChem ID
CID: 11584525
SID: 17155420
Canonical SMILES
CC1(C)C(C(=O)c2cn(CCN3CCOCC3)c3ccccc23)C1(C)C
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Compound Formula C22H30N2O2
Compound Structure
Protein Name
 Protein Info 
Cannabinoid receptor 1
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
>
Small molecule receptor (family A GPCR)
>
Lipid-like ligand receptor (family A GPCR)
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Cannabinoid receptor
Uniprot ID
P21554
Gene Name
CNR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  1
1
EC50 = 811 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 330 nM
2 Ki = 845 nM