Brief Information of the Compound and Protein
Compound Name
N-[1-(4-methoxy-2-methylphenyl)-3,6-dimethylpyrazolo[3,4-d]pyrimidin-4-yl]-5-(propylaminomethyl)-1,3,4-oxadiazol-2-amine
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PubChem ID
CID: 45485041
Canonical SMILES
CCCNCc1nnc(Nc2nc(C)nc3n(nc(C)c23)-c2ccc(OC)cc2C)o1
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Compound Formula C21H26N8O2
Compound Structure
Protein Name
Corticotropin-releasing factor receptor 1
Protein Classification
Membrane receptor
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Family B G protein-coupled receptor
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Peptide receptor (family B GPCR)
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Corticotropin releasing factor receptor
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Corticotropin releasing factor receptor
Uniprot ID
P34998
Gene Name
CRHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 996 nM
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