Brief Information of the Compound and Protein
Compound Name
1-(4-methoxy-2-methylphenyl)-3,6-dimethyl-N-(5-((propylamino)methyl)-1H-imidazol-1-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
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PubChem ID
CID: 45484976
Canonical SMILES
CCCNCc1cncn1Nc1nc(C)nc2n(nc(C)c12)-c1ccc(OC)cc1C
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Compound Formula C22H28N8O
Compound Structure
Protein Name
Corticotropin-releasing factor receptor 1
Protein Classification
Membrane receptor
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Family B G protein-coupled receptor
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Peptide receptor (family B GPCR)
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Corticotropin releasing factor receptor
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Corticotropin releasing factor receptor
Uniprot ID
P34998
Gene Name
CRHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 2500 nM
   TI
   LI
   LO
   TS