Brief Information of the Compound and Protein
Compound Name
 Compound Info 
N-[4-(3,4-dimethoxyphenyl)-4-[1,3-dioxo-4-[4-[(1R)-1-phenylethyl]piperazin-1-yl]isoindol-2-yl]butyl]thiophene-2-sulfonamide
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 PubChem ID
CID: 23627249
SID: 46488380
Canonical SMILES
COc1ccc(cc1OC)C(CCCNS(=O)(=O)c1cccs1)N1C(=O)c2cccc(N3CCN(CC3)[C@H](C)c3ccccc3)c2C1=O
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Compound Formula C36H40N4O6S2
Compound Structure
Protein Name
 Protein Info 
Urotensin-2 receptor
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
>
Peptide receptor (family A GPCR)
>
Short peptide receptor (family A GPCR)
>
Neuropeptide receptor
Uniprot ID
Q9UKP6
Gene Name
UTS2R
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000397 RMS13
 Cell Line Info 
Mus musculus (Mouse)  2
1
IC50 = 250 nM
   TI
   LI
   LO
   TS
2
Ki = 76 nM
   TI
   LI
   LO
   TS