Brief Information of the Compound and Protein
Compound Name
(4R,10bR)-4-(3,4-dimethoxyphenyl)-10-(4-ethylpiperazin-1-yl)-1,2,3,4-tetrahydropyrido[2,1-a]isoindol-6(10bH)-one
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PubChem ID
CID: 44206680
SID: 85206606
Canonical SMILES
CCN1CCN(CC1)c1cccc2C(=O)N3[C@H](CCC[C@@H]3c3ccc(OC)c(OC)c3)c12
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Compound Formula C26H33N3O3
Compound Structure
Protein Name
Urotensin-2 receptor
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
>
Peptide receptor (family A GPCR)
>
Short peptide receptor (family A GPCR)
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Neuropeptide receptor
Uniprot ID
Q9UKP6
Gene Name
UTS2R
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000397 RMS13 Mus musculus (Mouse)  1
1
Ki = 64 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 Ki = 64 nM