Brief Information of the Compound and Protein
Compound Name
1-Cyclopropyl-6-fluoro-4-oxo-7-(4-(4-(3-(piperidin-1-yl)propoxy)benzyl)piperazin-1-yl)-1,4-dihydroquinoline-3-carboxylic acid
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PubChem ID
CID: 46880384
Canonical SMILES
O=C(O)c1cn(C2CC2)c2cc(N3CCN(Cc4ccc(OCCCN5CCCCC5)cc4)CC3)c(F)cc2c1=O
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Compound Formula C32H39FN4O4
Compound Structure
Protein Name
Histamine H3 receptor
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Histamine receptor
Uniprot ID
Q9Y5N1
Gene Name
HRH3
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
Ki = 1.995 nM
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