Brief Information of the Compound and Protein
Compound Name
(-)-Dimethyl-{2-[3-((R)-1-pyrazin-2-yl-ethyl)-1H-inden-2-yl]-ethyl}-amine
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PubChem ID
CID: 44247806
SID: 85281510
Canonical SMILES
C[C@H](C1=C(CCN(C)C)Cc2ccccc12)c1cnccn1
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Compound Formula C19H23N3
Compound Structure
Protein Name
Histamine H1 receptor
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Histamine receptor
Uniprot ID
P35367
Gene Name
HRH1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000386 Flp-In-CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 1.3 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 Ki = 1.3 nM
2 Ki = 1.5 nM