Brief Information of the Compound and Protein
Compound Name
(1R,5S)-9-Bromo-1,2,3,4,5,6-hexahydro-1,5-methano-pyrido[1,2-a][1,5]diazocin-8-one
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PubChem ID
CID: 15519735
Canonical SMILES
O=c1c(Br)ccc2n1C[C@@H]1CNC[C@H]2C1
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Compound Formula C11H13BrN2O
Compound Structure
Protein Name
Neuronal acetylcholine receptor subunit alpha-3
Protein Classification
Ion channel
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Ligand-gated ion channel
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Nicotinic acetylcholine receptor
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Nicotinic acetylcholine receptor alpha subunit
Uniprot ID
P32297
Gene Name
CHRNA3
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000016 IMR-32 Homo sapiens (Human)  1
1
IC50 = 15.6 nM
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