Brief Information of the Compound and Protein
Compound Name
 Compound Info 
3-Cyclohexyl-1-[4'-((3R,5S)-3,5-dimethyl-piperazin-1-ylmethyl)-biphenyl-2-ylmethyl]-1-[2-(3-methoxy-phenyl)-ethyl]-urea
    Show/Hide
 PubChem ID
CID: 16752689
SID: 57248732
Canonical SMILES
COc1cccc(CCN(Cc2ccccc2-c2ccc(CN3C[C@H](C)N[C@H](C)C3)cc2)C(=O)NC2CCCCC2)c1
    Show/Hide
Compound Formula C36H48N4O2
Compound Structure
Protein Name
 Protein Info 
Motilin receptor
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
>
Peptide receptor (family A GPCR)
>
Short peptide receptor (family A GPCR)
>
Motilin receptor
Uniprot ID
O43193
Gene Name
MLNR
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  1
1
EC50 = 10 nM
   TI
   LI
   LO
   TS
CL000006 HEK293
 Cell Line Info 
Homo sapiens (Human)  1
1
EC50 = 50.12 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 EC50 = 10 nM