Brief Information of the Compound and Protein
Compound Name
3-[3-methoxy-4-(2-pyrrolidin-1-ylethoxy)phenyl]-6-[4-(trifluoromethyl)phenyl]thieno[3,2-d]pyrimidin-4-one
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PubChem ID
CID: 44416337
Canonical SMILES
COc1cc(ccc1OCCN1CCCC1)-n1cnc2cc(sc2c1=O)-c1ccc(cc1)C(F)(F)F
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Compound Formula C26H24F3N3O3S
Compound Structure
Protein Name
Melanin-concentrating hormone receptor 1
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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MCH receptor
Uniprot ID
Q99705
Gene Name
MCHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
IC50 = 2.512 nM
   TI
   LI
   LO
   TS