Brief Information of the Compound and Protein
Compound Name
 Compound Info 
(R)-5-chloro-6-(4-(4-(4-fluorophenyl)-6-(trifluoromethyl)-1Hbenzo[d]imidazol-2-yl)-3-methylpiperazin-1-yl)pyridin-3-amine
    Show/Hide
 PubChem ID
CID: 11634799
SID: 16737951
Canonical SMILES
C[C@@H]1CN(CCN1c1nc2c(cc(cc2[nH]1)C(F)(F)F)-c1ccc(F)cc1)c1ncc(N)cc1Cl
    Show/Hide
Compound Formula C24H21ClF4N6
Compound Structure
Protein Name
 Protein Info 
Transient receptor potential cation channel subfamily V member 1
Protein Classification
Ion channel
>
Voltage-gated ion channel
>
Transient receptor potential channel
Uniprot ID
O35433
Gene Name
TRPV1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  2
1
IC50 = 33 nM
   TI
   LI
   LO
   TS
2
IC50 = 98 nM
   TI
   LI
   LO
   TS