Brief Information of the Compound and Protein
Compound Name
 Compound Info 
2-(4-(trifluoromethyl)phenyl)-6-(3-(trifluoromethyl)pyridin-2-yl)-1,2,4,5,6,7-hexahydropyrazolo[3,4-b]pyridin-3-one
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Canonical SMILES
Oc1c2c(nn1-c1ccc(C(F)(F)F)cc1)NC(c1ncccc1C(F)(F)F)CC2
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Compound Formula C19H14F6N4O
Compound Structure
Protein Name
 Protein Info 
Transient receptor potential cation channel subfamily V member 1
Protein Classification
Ion channel
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Voltage-gated ion channel
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Transient receptor potential channel
Uniprot ID
Q8NER1
Gene Name
TRPV1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  1
1
IC50 = 290 nM
   TI
   LI
   LO
   TS