Brief Information of the Compound and Protein
Compound Name
N-[3-[4-[6-[(4-methylpiperazin-1-yl)methyl]-1,4-dihydroindeno[1,2-c]pyrazol-3-yl]thiophen-2-yl]prop-2-ynyl]benzenesulfonamide
    Show/Hide
PubChem ID
CID: 16221258
SID: 24903733
Canonical SMILES
CN1CCN(Cc2ccc-3c(Cc4c-3n[nH]c4-c3csc(c3)C#CCNS(=O)(=O)c3ccccc3)c2)CC1
    Show/Hide
Compound Formula C29H29N5O2S2
Compound Structure
Protein Name
Potassium voltage-gated channel subfamily H member 2
Protein Classification
Ion channel
>
Voltage-gated ion channel
>
Potassium channels
>
Voltage-gated potassium channel
Uniprot ID
Q12809
Gene Name
KCNH2
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 4870 nM
   TI
   LI
   LO
   TS