Brief Information of the Compound and Protein
Compound Name
1-(5-((2H-tetrazol-5-yl)carbamoyl)-2,3-dihydro-1H-inden-1-yl)-1-(cis-4-tert-butylcyclohexyl)-3-(4-(trifluoromethoxy)phenyl)urea
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Canonical SMILES
CC(C)(C)[C@@H]1CC[C@@H](CC1)N(C1CCc2cc(ccc12)C(=O)Nc1nnn[nH]1)C(=O)Nc1ccc(OC(F)(F)F)cc1
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Compound Formula C29H34F3N7O3
Compound Structure
Protein Name
Gastric inhibitory polypeptide receptor
Protein Classification
Membrane receptor
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Family B G protein-coupled receptor
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Peptide receptor (family B GPCR)
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Glucagon-like receptor
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Gastric inhibitory polypeptide receptor
Uniprot ID
P48546
Gene Name
GIPR
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
IC50 = 435 nM
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