Brief Information of the Compound and Protein
Compound Name
(2R)-3-(1H-indol-3-yl)-N-(2-phenylethyl)-2-[[[2-(1,2,3,4-tetrahydroisoquinolin-1-yl)acetyl]amino]carbamoylamino]propanamide
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PubChem ID
CID: 44387452
Canonical SMILES
O=C(CC1NCCc2ccccc12)NNC(=O)N[C@H](Cc1c[nH]c2ccccc12)C(=O)NCCc1ccccc1
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Compound Formula C31H34N6O3
Compound Structure
Protein Name
Bombesin receptor subtype-3
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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GRP-related receptor
Uniprot ID
P32247
Gene Name
BRS3
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
EC50 = 19 nM
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