Brief Information of the Compound and Protein
Compound Name
 Compound Info 
4'-Oxazol-2-yl-2'-pyrazol-1-ylmethyl-biphenyl-2-sulfonic acid (3,4-dimethyl-isoxazol-5-yl)-amide
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 PubChem ID
CID: 11730445
SID: 16836226
Canonical SMILES
Cc1noc(NS(=O)(=O)c2ccccc2-c2ccc(cc2Cn2cccn2)-c2ncco2)c1C
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Compound Formula C24H21N5O4S
Compound Structure
Protein Name
 Protein Info 
Endothelin-1 receptor
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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Endothelin receptor
Uniprot ID
P25101
Gene Name
EDNRA
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  1
1
Ki = 0.3 nM
   TI
   LI
   LO
   TS