Brief Information of the Compound and Protein
Compound Name
N-(2,6-dimethylphenyl)-5-[5-(4-methylpiperazin-1-ylmethyl)thiophen-2-yl]imidazo[1,5-a]pyrazin-8-amine hydrochloride
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PubChem ID
CID: 118725186
Canonical SMILES
Cc1cccc(C)c1Nc1ncc(-c2ccc(CN3CCCC3)s2)n2cncc12.Cl
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Compound Formula C23H26ClN5S
Compound Structure
Protein Name
Proto-oncogene tyrosine-protein kinase Src
Protein Classification
Enzyme
>
Kinase
>
Protein Kinase
>
TK protein kinase group
>
Tyrosine protein kinase Src family
Uniprot ID
P12931
Gene Name
SRC
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000053 COS-7 Chlorocebus aethiops (Green monkey)  1
1
IC50 = 820 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 52 nM