Brief Information of the Compound and Protein
Compound Name
3-(2,6-dichloropyridin-4-yl)-1-((3R,6S)-6-(3-((dimethylamino)methyl)phenyl)bicyclo[4.1.0]heptan-3-yl)-1-((1-(methylsulfonyl)piperidin-4-yl)methyl)urea
    Show/Hide
PubChem ID
CID: 44424258
Canonical SMILES
CN(C)Cc1cccc(c1)[C@@]12CC1C[C@@H](CC2)N(CC1CCN(CC1)S(C)(=O)=O)C(=O)Nc1cc(Cl)nc(Cl)c1
    Show/Hide
Compound Formula C29H39Cl2N5O3S
Compound Structure
Protein Name
Melanin-concentrating hormone receptor 1
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
>
Peptide receptor (family A GPCR)
>
Short peptide receptor (family A GPCR)
>
MCH receptor
Uniprot ID
Q99705
Gene Name
MCHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 3.3 nM
   TI
   LI
   LO
   TS