Brief Information of the Compound and Protein
Compound Name
(E)-N-(4,5-dichlorothiophen-2-yl)sulfonyl-3-[1-[(3-methoxyphenyl)methyl]-3a-methyl-2-oxo-3,4,5,6-tetrahydroindol-7-yl]prop-2-enamide
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PubChem ID
CID: 44571291
Canonical SMILES
COc1cccc(CN2C(=O)CC3(C)CCCC(\C=C\C(=O)NS(=O)(=O)c4cc(Cl)c(Cl)s4)=C23)c1
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Compound Formula C24H24Cl2N2O5S2
Compound Structure
Protein Name
Prostaglandin E2 receptor EP3 subtype
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Lipid-like ligand receptor (family A GPCR)
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Prostanoid receptor
Uniprot ID
P43115
Gene Name
PTGER3
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000026 CHO-K1 Cricetulus griseus (Chinese hamster)  1
1
IC50 = 5.8 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 6.4 nM